• Synthesis and application of phosphonothioates, phosphonodithioates, phosphorothioates, phosphinothioates and related compounds 

  Jones, David J.; O'Leary, Eileen M.; O'Sullivan, Timothy P. (Elsevier, 2018-10-26)

  Methods for the preparation of phosphonothioates, phosphonodithioates, phosphorothioates, phosphinothioates and related compounds are reviewed. The application of these compounds as synthetic intermediates is also discussed.
• Synthetic and stereochemical aspects of enantioselective copper catalysed C-H insertion reactions leading to cyclopentanones and sultones 

  Shiely, Amy E. (University College Cork, 2018)

  This thesis describes the synthesis of a series of α-diazocarbonyl compounds including α-diazoβ-keto sulfones, α-diazo-β-keto phosphine oxides, 2-diazo-1,3-diketones and αdiazosulfonates, and their reactivity in intramolecular ...
• Synthesis of novel quinine analogs and evaluation of their effects on Trypanosoma cruzi 

  Ceole, Ligia F.; Gandhi, Hirenkumar; Villamizar, Luz H.; Soares, Maurilio J.; O'Sullivan, Timothy P. (Future Science: Newlands Press, 2018-02)

  Aim: Chagas disease is a tropical disease caused by the hemoflagellate protozoan Trypanosoma cruzi. There is no vaccine for Chagas disease and available drugs (e.g., benznidazole) are effective only during the acute phase, ...
• Asymmetric peroxidation of α,β-unsaturated aldehydes under diarylprolinol ether catalysis 

  O'Reilly, Kate; Gupta, Manoj K.; Gandhi, Hirenkumar; Kumar, Vydyula P.; O'Sullivan, Timothy P. (Bentham Science Publishers, 2017)

  Background: Chiral peroxides, many of which are biologically active, are an attractive target in organic synthesis. Organocatalysts have been used for some time in the asymmetric epoxidation of α,β- unsaturated carbonyls. ...
• Preparation of γ,δ-unsaturated-β-ketoesters: Lewis acid-catalysed CH insertion of ethyl diazoacetate into α,β-unsaturated aldehydes 

  Gandhi, Hirenkumar; O'Sullivan, Timothy P. (Elsevier, 2017-07-29)

  The synthesis of γ,δ-unsaturated-β-keto esters was achieved by the Lewis acid-catalysed direct CH insertion of an α-diazoester into various α,β-substituted-unsaturated aldehydes. CH insertion of ethyl diazoacetate into ...

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